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Adrenergic System (Sympathetic)

Adrenergic Agonist Direct (Ep,NEp)


-Ergotamine -Oxymetazoline 1 -Phenylpropanolamine 1 -Phenylephrine 1 -Clonidine 2 -Methyldopa 2 -Guanfacin 2

Adrenergic Antagonist (Blockers)


(Labetolol)

Indirect
(Sympathomimetic)

-Isoprotrenol 1,2 -Dobutamine 1 -Albuterol 2 -Terbutaline 2 -Metoprotrenol 2

-Tyramine -Phenoxybenzamine 1,2 -Ephidrine -Phentolamine 1,2 -Amphetamine -Prazocin 1 -Tolazoline 2 - Yohimbine 2

(lol)
-Propranolol 1,2 -Timolol 1,2 -Acetbutolol 1 -Atenolol 1 -Betaxolol 1 -Metoprolol 1

Cholinergic System (Parasympathetic)


Cholinergic Agonist Direct Indirect (AchE inhibitors) Reversible
-Ach -Methacholine -Bethanechol -Pilocarpine -Physostigmine -Neostigmine -Pyridostigmine

Cholinergic Antagonist
(Antimuscarinic,Antinicotinic)

Irreversible
-Organophosphate esters (Insecticide, Nerve gases) e.g.-Isoflurophate -Ecothiophate -Malathione -Atropine -Scopolamine -Trihexaphenidyl -Ipratropium -Glycopyrrolate -Propantheline -Benzatropine -Dicyclomine -Pirenzepine -Mecamylamine -Trimethaphan -Hexamethonium

Quaternary nitrogen Tertiary nitrogen Ganglionic blockers

Neuromuscular blockers
Nondepolarizing (Competitive drugs)
-X-curarine e.g.-Tubocurarine -X-curonium -X-curium -Gallamine

Depolarizing (Noncompetitive drugs)


-Succinylcholine

Done by Dr. AhmeDSh unDer SuperviSion of Dr.yAyoo

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