Endocrine pharmacology

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1. GH analogs Somatropin, somatrem 21. Progestin (partial Danazole (do not confuce with
agonist ) aromatase inhibitors)
2. Somatostatin Ocreotide
analog 22. Antiprogestin Mifepristone (RU 486)
3. ACTH analog Cosytropin 23. Androgens Methyltestosterone, fluoxymesterone
(synthetic)
4. GnRH receptor Leuprolide
agonist 24. Androgens Oxandrolone, stanozolol
(anabolic)
5. FSH analog Urofollitropin, follitropin alpha
25. Androgen Flutamide, bicalutamide
6. LH analog hCG
receptor
7. FSH plus LH Menotropins antagonists
activity
26. 5-alpha-reductase Finasteride
8. Prolactin-release Bromocriptine (dopamine analog), inhibitor
inhibitors pergolide, cabergoline
27. Androgen Ketoconazole
9. Vasopressin Desmopressin synthesis inhibitor
analog
28. Ultra-rapid-acting Lispro
10. Antithyroid drugs 1. Thioamides: PTU and methimazole insulin
(block iodination and possibly MIT-DIT
29. Rapid-actin insulin Human crystalline insulin
coupling)
2. Iodide salts 30. Intermediate- NPH (isophane), Lente
3. Radioactive iodine (I-131) acting insulin
4. Propranolol
31. Long-acting Ultralente
5. Ipodate
insulin
11. Glucocorticoid Prednisolone, triamcinolone,
32. Ultra-long-acting Glargine
agonists dexamethasone (increasing degree of
duration, anti-inflammatory effect and 33. GLP-1 analogs Sitagliptin, exenatide
topical activity) 34. Insulin 1. Sulfonylureas: glipizide, glimepiride,
Betamethasone is given to pregnant secretagogues glyburide (2nd gen) and
women to boost surfactant production chlorpropamide, tolbutamide (1st gen)
in the fetus 2. Meglitinides: repaglinide
12. Glucocorticoid Mifepristone 3. Nateglinide
receptor 35. Biguanides Metformin
antagonists
36. Thiazolidinediones Pioglitazone, rosiglitazone
13. Glucocorticoid Ketoconazole, aminoglutethimide,
37. alpha-glucosidase Acarbose, miglitol
synthesis metyrapone
inhibitors
inhibitors
38. Bisphosphonates Older: Etidronate, pamidronate (<12
14. Mineralocorticoids Fludrocortisone (long duration of
months)
action)
Newer: Alendronate, risedronate (>5 yrs)
15. Mineralocorticoid Spironolactone, eplerenone
39. RANKL-inhibitor Denosumab
receptor inhibitors
40. Calcium mimetic Cinacalcet
16. Estrogens Estradiol, estriol, estrone
(natural) 41. Serum calcium Plicamycin, mithramycin
reducer
17. Estrogens Ethinyl estradiol, mestranol,
(antibiotic)
(synthetic) diethylstilbestrol
18. SERMs Tamoxifen and raloxifene. Clomiphene.
19. Aromatase Anastrozole, letrozole
inhibitors
20. Progestins Norgestrel, medoxyprogesterone,
(synthetic) norgestimate, norethindrone