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2. ANTI-INFECTIVE AGENTS 8
2.1 AMEBICIDES ………………………………………………………………………..………8
2.2 ANTHELMINTICS ………………………………………………………....…….…….……9
2.3 ANTIBIOTICS ………………………………………………………………...…………… 11
2.3.1 ANTIFUNGAL ANTIBIOTICS ………………………………………………… 11
2.3.2 AMINOGLYCOSIDES ……………………………………………….………... 17
2.3.3 CEPHALOSPORINS ……………………………………………………….…. 20
2.3.3.1 FIRST GENERATION CEPHALOSPORINS …………….……….. 21
2.3.3.2 SECOND GENERATION CEPHALOSPORINS ………………….. 22
2.3.3.3 THIRD GENERATION CEPHALOSPORINS ……………...……… 25
2.3.3.4 FOURTH GENERATION CEPHALOSPORINS ………………….. 29
2.3.4 CHLORAMPHENICOLS ………………………………………………….…... 30
2.3.5 MACROLIDES ………………………………………………….………………31
2.3.6 PENICILLINS ……………………………………………………….……...….. 33
2.3.6.1 NATURAL PENICILLINS ………………………………….………… 34
2.3.6.2 PENICILLINASE-RESISTANT PENICILLINS…….………………. 35
2.3.6.3 AMINOPENICILLINS ………………………………………….…….. 36
2.3.6.4 EXTENDED-SPECTRUM PENICILLINS….…………………..…… 40
2.3.7 TETRACYCLINES ……………………………………………………………. 40
2.3.7.1 LONG-ACTING TETRACYCLINES ..……………….……………… 41
2.3.8 MISCELLANEOUS ANTIBIOTICS …………………………………….…….. 42
2.4 ANTITUBERCULOSIS AGENTS ………………………………………………….……. 48
2.5 ANTIVIRALS …………………………………………………………………….………… 50
2.6 ANTIMALARIALS ………………………………………………………………………….65
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3. ANTINEOPLASTIC AGENTS 77
3.1 ALKYLATING AGENTS ………………………………………………….………………. 77
3.2 ANTIMETABOLITES ………………………………………………………….………….. 85
3.3 CYTOTOXIC ANTIBIOTICS AND RELATED SUBTANCES……..…….……………..93
3.4 PLANT ALKALOIDS AND OTHER NATURAL PRODUCTS….…….…..…......…… 100
3.5 HORMONES………………………….........……………………………………...…….. 108
3.5.1 ANTIANDROGENS……………………………………….......….………..… 108
3.5.2 ANTIESTROGENS……………………..…………………...……………..… 108
3.5.3 AROMATASE INHIBITORS.……………………………………...……….... 109
3.5.4 GONADOTROPIN RELEASING HORMONE AND RELATED
SYNTHETIC DRUGS………………………………………………………… 111
3.5.5 PROGESTINS ………………...……………………………………...……… 115
3.6 MONOLCLNAL ANTIBODIES……………………...……………….………......…....... 116
3.7 TYROSINE KINASE INHIBITORS………………………………………………...……119
3.8 OTHER ANTINEOPLASTIC AGENTS………………………………………………… 121
3.9 ANTINEOPLASTIC ADJUNCTS……………………………………………….………. 126
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บัญชียาสมุนไพร……………………………………………………………..……………..…………… 499
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