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MACP 2113
Disediakan oleh:
Pengajar U41
Kolej Pembantu Perubatan, Ulu Kinta
OBJEKT
IF
1. Memberi definisi ubatan
antibiotik topikal.
2. Menyatakan tujuan/ indikasi ubat.
3. Menyatakan dos dan contoh ubat.
Antibiotik
Topikal
Antibiotik topikal
Adalah ubat yang
digunakan untuk merawat
jangkitan bakteria topikal
(luaran).
Tindakan
Bacteriostatic (menghalang
pembiakan/ pertumbuhan
bakteria)
Bactericidal (membunuh
bakteria)
Contoh
ubat
chloramphenicol
(Chloromycetin)
chlortetracycline
(Aureomycin)
neomycin (Neosporin)
gentamycin (Garamycin)
sulphacetamide (Albucid)
1. chloramphenicol
(Chloromycetin 0.5% Eye Drop)
Category: C
Broad spectrum.
Bacteriostatic (prevent cell
replication)
Mudah diserap ke dalam mata.
Indication
Bacterial infection of the
eye
Konjunctivitis - semua
peringkat umur
Blepharitis
Abrasi kornea - pencegahan
Dose
1-2 drops every 3-4 hours
Reduce frequency (once
infection is controlled)
Continue for 48 hour after
healing (1-2 drops qid)
2. chloramphenicol
(Chloromycetin 1% Eye Oinment)
Category: C
Broad spectrum.
Bacteriostatic (prevent cell
replication)
Mudah diserap ke dalam mata.
Indication
Bacterial infection of the eye
Konjunctivitis - semua
peringkat umur
Blepharitis
Abrasi kornea - pencegahan
Dose
Apply of ointment into
conjunctival sac at night (if
eye drops used during day
time) or
Apply of ointment into
conjunctival sac tid-qid (if
eye oinment used alone)
Kesan sampingan
Allergic
Irritation, burning, itching, urticaria
Superinfection
Bone marrow hypoplasia (long
term)
Aplastic anemia (long term)
Contraindication
Allergic to chloramphenicol
Cautious
3. chlortetracycline
(Aureomycin 1% Eye Oinment)
Category: B
Broad spectrum.
Bacteriostatic
Berkesan terhadap organisma
Gram +ve dan Gram ve.
Indication
Superficial bacterial infection
of the eye (gram +ve & -ve
including trachoma)
Eyelid infection
Dose
Apply 1 drop tid-qid (if eye
oinment used alone)
Kesan sampingan
Allergic
Irritation, burning, itching, urticaria
Superinfection
Contraindication
Allergic to chlortetracycline
4. neomycin
(Neosporin Eye Drop)
Category: B
Indication
Superficial bacterial infection
of the eye (gram -ve)
Dose
1-2 drops bid-qid
Severe infection: 1-2 drops
every 15-30 mins
Kesan
Sampingan
Urticaria
Itching
Irritation
Pain
Dermatitis
Rash
Contraindication
Allergic to neomycin
Pregnancy
Lactation
5. gentamycin
(Garamycin 0.3% Eye Drop)
Category: A
Indication
Superficial bacterial
infection of the eye
(Pseudomonas aeruginosa)
Dose
1-2 drops bid-qid
6. Gentamycin
(Garamycin Eye Oinment)
Category: A
Indication
Superficial bacterial infection
of the eye (Pseudomonas
aeruginosa)
Dose
Apply into the conjunctival
sac tid-qid
Kesan
Sampingan
Transient irritation
Burning
Stinging
Itching
Dermatitis
Superinfection
Contraindication
Allergic to gentamycin
Cautious
Contact lens users
Pregnancy
Lactation
7. sulphacetamide
(Albucid 10% Eye Drop)
Category: B
Bakteriostatik
Indication
Mild infection of conjunctiva
Eyelid infection
Industrial eye injuries
Dose
Apply 1-2 drops every 2-6
hours
Kesan
Sampingan
Iritation
Itching
Dermatitis
Contraindication
Allergic to sulphacetamide
Interactions
Not found
Anti-Viral
Topikal
Antibiotik topikal
Adalah ubat yang
digunakan untuk
merawat jangkitan virus
pada mata.
Tindakan
Interferes with viral
reproduction by altering DNA
synthesis.
Contoh
ubat
acyclovir (Zovirax)
1. acyclovir
(Zovirax 3% Eye Oinment)
Category: A*
Indication
Herpes Simplex
keratitis
Dose
Applied 1cm into conjunctival
sac 5 times/day.
Continue for about 3 days
after healing.
Kesan
Sampingan
Iritation
Inflammation
Edema of eyelids
Allergic reactions
photophobia
Contraindication
Allergic to drugs
Interactions
Not found
1.
Soala
n
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