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GOUT
Dr.dr. Asep Sukohar, M.Kes
Bagian Farmakologi dan Terapi FK Unila
Metabolisme asam urat, enzim dan mekanisme obat
Gout is a form of arthritis in which
uric acid accumulates in increased
amounts in the blood and often is
deposited in the joints.
Colchicine
• nausea, vomiting, diarrhea, abdominal pain, and bone
marrow depression
Probenecid
• headache, GI symptoms, urinary frequency, and
hypersensitivity reactions.
Sulfinpyrazone
• Gastrointestinal disturbances
Allopurinol Colchicine Probenecid Sulfinpyrazon